Drug Action/uses | Drug |
Cholinergic agonist, stereochemical centre, negative isomer lacks affinity | |
Adenosine Receptor Agonist | |
Causes permenant activation of Adenylyl Cyclase | |
Anti diabetic drug that inhibits ATP sensitive K+ channels, leading to membrane depolarization | |
Glucocortisol agonist, labour inducing agent | |
Calcium agonist (L, T, N VGCC). Dihydropiridine, therefore lipid soluble | |
beta adrenoreceptor agonist, used in bradycardia | |
Muscarinic Ach Receptor Antagonist | |
Progesterone agonist. Inhibits ovarian steroidogenesis | |
Potassium channel opener (hyperpolarizes cell via efflux of K+ ions, causes vasodilation) | |
Classic DHP, VGCC blocker | |
Irreversable Muscarinic Ach antagonist | |
Glucocorticoid agonist used in autoimmune conditions (canker in horses) | |
Ester type local anaesthetic. NA+ channel blocker, weak base-has to enter cell. | |
Blocks NaV 1.8 and 1.9 (uncharged, hydrophobic) | |
Slow in-slow out Local Anaesthetic, use dependant at low concs | |
Progesterone receptor agonist | |
Antagonist to nicotinic Ach receptor, binds competitively and irreversibly. Cannot cross BBB | |