Activates alpha and beta receptors
Activates alpha-1 receptors
Activates alpha-2 receptors
Activates benzodiazepine receptor
Activates beta-1 receptors
Activates beta-2 receptors
Activates cGMP
Activates cholinergic receptors
Activates dopamine receptors
Activates Gaba Receptor
Activates muscarinic receptor
Binds alpha subunit of benzodiazepine receptor
Binds phencyclidine receptor to inhibit glutamate
Blocks alpha-1 & 2 receptor
Blocks alpha-1 receptor
Blocks alpha-1, beta-1 & 2 receptors
Blocks angiotensin II receptor
Blocks benzodiazepine receptor
Blocks beta-1 receptor
Blocks endothelin receptors
Blocks Na+ channels
Ca++ channel blocker
Depletes NE from presynaptic site
Depolarizing nicotinic receptor blocker
Directly inhibits renin
Gaba agonist
Induce NE release
Inhibits aldehyde dehydrogenase
Inhibits ACh release
Inhibits ACh-Esterase
Inhibits alcohol dehydrogenase
Inhibits angiotensin converting enzyme
Inhibits glutaminergic/activates gabaergic neurons
Inhibits NE reuptake
Inhibits release of Ca++
Inhibits tyrosine hydroxylase
Irreversibly blocks Na+ channels
Irreversibly inhibits ACh-Esterase
Non-depolarizing nicotinic receptor blocker
Opens K+ channels in s.m.
Partial 5HT agonist
Reversibly blocks muscarinic receptor
Activate opiate receptor/block 5HT reuptake
Activates Gaba
Activates GnRH receptor
Alkylating agent
Bind ergosterol
Bind THC receptor
Bind to a receptor to increase lipocortin
Bind to opiate receptors
Binds 30s & inhibits tRNA binding
Binds 50s & inhibits translocation
Binds adenosine receptor
Binds bacterial isoleucyl tRNA synthetase
Binds bile acids
Binds CD20
Binds dialanine residues
Binds fungal microtubules
Binds HER2
Binds PPAR
Binds TNF
Binds to & inhibits CD80 & CD86 receptors
Binds to alpha integrins on CD4 T cells
Binds to antithrombin 3
Binds to cyclophyllin to inhibit enzyme
Binds to FKBP to inhibit enzyme
Binds to IL-1 molecule
Binds to IL-12 & IL-23
Binds to IL-6 receptors
Binds to microtubules
Binds to mRNA for apolipoprotein B
Binds to negatively charged sites on LPS
Binds to PBP
Binds to virus to inhibit fusion
Block dopamine receptors w/ high affinity
Block dopamine/histamine/5HT receptors
Block H1 receptors
Block H2 receptors
Block leukotriene receptors
Blocks androgen receptor
Blocks binding site on macrophage
Blocks cholesterol transporters
Blocks cholesterol uptake
Blocks estrogen receptor
Blocks fusion of virus w/ target cell
Blocks H+ channel in endosome
Blocks IL-2 receptor
Blocks synth of NAM
Blocks VEGF
Causes strand breakage
Cholinergic reuptake inhibitor
COMT inhibitor
Converted to free radical
Converts plasminogen to plasmin
Decreases platelet formation
Directly activate dopamine receptors
Directly inhibits thrombin
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